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Enzymatic Transition States and Drug Design

Transition state theory teaches that chemically stable mimics of enzymatic transition states will bind tightly to their cognate enzymes. Kinetic isotope effects combined with computational quantum chemistry provides enzymatic transition state information with sufficient fidelity to design transition...

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Dades bibliogràfiques
Publicat a:Chem Rev
Autor principal: Schramm, Vern L.
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6615489/
https://ncbi.nlm.nih.gov/pubmed/30335982
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.chemrev.8b00369
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