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Benzimidazoles Downregulate Mdm2 and MdmX and Activate p53 in MdmX Overexpressing Tumor Cells

Tumor suppressor p53 is mutated in about 50% of cancers. Most malignant melanomas carry wild-type p53, but p53 activity is often inhibited due to overexpression of its negative regulators Mdm2 or MdmX. We performed high throughput screening of 2448 compounds on A375 cells carrying p53 activity lucif...

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Dettagli Bibliografici
Pubblicato in:Molecules
Autori principali: Mrkvová, Zuzana, Uldrijan, Stjepan, Pombinho, Antonio, Bartůněk, Petr, Slaninová, Iva
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6600429/
https://ncbi.nlm.nih.gov/pubmed/31181622
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24112152
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