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Design, synthesis and evaluation of [(111)In]-labeled, DOTA-conjugated tetrapeptides having high affinity and selectivity for mu opioid receptors

INTRODUCTION: Peripheral mu (μ) opioid receptors are implicated in pain, bowel dysfunction and the progression of certain cancers. In an effort to identify radioligands well suited for imaging these peripheral sites, we have prepared and evaluated four hydrophilic [(111)In]-labeled, DOTA (1,4,7,10-t...

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Detalles Bibliográficos
Publicado en:Nucl Med Biol
Main Authors: Lever, John R., Fergason-Cantrell, Emily A., Carmack, Terry L., Watkinson, Lisa D., Gallazzi, Fabio
Formato: Artigo
Idioma:Inglês
Publicado: 2019
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6591026/
https://ncbi.nlm.nih.gov/pubmed/30933866
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nucmedbio.2019.02.001
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