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Effect of DOTA Position on Melanoma Targeting and Pharmacokinetic Properties of (111)In-labeled Lactam Bridge-Cyclized Alpha-Melanocyte Stimulating Hormone Peptide

The purpose of this study was to examine the effect of DOTA (1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid) position on melanoma targeting and pharmacokinetics of radiolabeled lactam bridge-cyclized alpha-melanocyte stimulating hormone (α-MSH) peptide. METHOD: A novel lactam bridge-cycliz...

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Autori principali: Guo, Haixun, Yang, Jianquan, Gallazzi, Fabio, Prossnitz, Eric R., Sklar, Larry A., Miao, Yubin
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2786309/
https://ncbi.nlm.nih.gov/pubmed/19817405
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bc9003475
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