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Cereblon versus VHL: Hijacking E3 ligases against each other using PROTACs

The von Hippel-Lindau (VHL) and cereblon (CRBN) proteins are substrate recognition subunits of two ubiquitously expressed and biologically important Cullin RING E3 ubiquitin ligase complexes. VHL and CRBN are also the two most popular E3 ligases being recruited by bifunctional Proteolysis-targeting...

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Dades bibliogràfiques
Publicat a:Bioorg Med Chem
Autors principals: Girardini, Miriam, Maniaci, Chiara, Hughes, Scott J., Testa, Andrea, Ciulli, Alessio
Format: Artigo
Idioma:Inglês
Publicat: Elsevier Science 2019
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6561380/
https://ncbi.nlm.nih.gov/pubmed/30826187
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2019.02.048
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