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Genetics and mechanisms of NT5C2-driven chemotherapy resistance in relapsed ALL

Mutations in the cytosolic 5′ nucleotidase II (NT5C2) gene drive resistance to thiopurine chemotherapy in relapsed acute lymphoblastic leukemia (ALL). Mechanistically, NT5C2 mutant proteins have increased nucleotidase activity as a result of altered activating and autoregulatory switch-off mechanism...

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Detaylı Bibliyografya
Yayımlandı:Blood
Asıl Yazarlar: Dieck, Chelsea L., Ferrando, Adolfo
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: American Society of Hematology 2019
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6533602/
https://ncbi.nlm.nih.gov/pubmed/30910786
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2019-01-852392
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