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Lead optimization of selective tubulin inhibitors as anti-trypanosomal agents

Previously synthesized tubulin inhibitors showed promising in vitro selectivity and activity against Human African Trypanosomiasis. Current aim is to improve the ligand efficiency and reduce overall hydrophobicity of the compounds, by lead optimization. Via combinatorial chemistry, 60 new analogs we...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Zhao, Anran, Li, Yaxin, Orahoske, Cody M., Schnur, Brittny, Sabbagh, Abboud, Zhang, Wenjing, Li, Bibo, Su, Bin
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6531046/
https://ncbi.nlm.nih.gov/pubmed/30833159
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2019.02.049
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