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Probing Structure-Activity Relationship in β-Arrestin2 Recruitment of Diversely Substituted Adenosine Derivatives

In the adenosine receptor (AR) subfamily of G protein-coupled receptors (GPCRs), biased agonism has been described for the human A(1)AR, A(2B)AR and A(3)AR. While diverse A(3)AR agonists have been evaluated for receptor binding and Gi-mediated cAMP signalling, the β-arrestin2 (βarr2) pathway has bee...

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Vydáno v:Biochem Pharmacol
Hlavní autoři: Storme, Jolien, Tosh, Dilip K., Gao, Zhan-Guo, Jacobson, Kenneth A., Stove, Christophe P.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6530469/
https://ncbi.nlm.nih.gov/pubmed/30292756
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2018.10.003
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