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Quantitative Ranking of Ligand Binding Kinetics with a Multiscale Milestoning Simulation Approach

Efficient prediction and ranking of small molecule binders by their kinetic (k(on) and k(off)) and thermodynamic (∆tt) properties can be a valuable metric for drug lead optimization, as these quantities are often indicators of in vivo efficacy. We have previously described a hybrid molecular dynamic...

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Vydáno v:J Phys Chem Lett
Hlavní autoři: Jagger, Benjamin R., Lee, Christopher T., Amaro, Rommie E.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6443090/
https://ncbi.nlm.nih.gov/pubmed/30070844
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jpclett.8b02047
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