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MEK drives BRAF activation through allosteric control of KSR proteins

RAF family kinases play prominent roles in cancer(1). Their activation is dependent on dimerization of their kinase domains, which has emerged as a roadblock for drug development(2,3). In mammals, RAF family kinases include three catalytically competent enzymes (A, B, and CRAF) and two pseudokinases...

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Publicado en:Nature
Autores principales: Lavoie, Hugo, Sahmi, Malha, Maisonneuve, Pierre, Marullo, Sara A., Thevakumaran, Neroshan, Jin, Ting, Kurinov, Igor, Sicheri, Frank, Therrien, Marc
Formato: Artigo
Lenguaje:Inglês
Publicado: 2018
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6433120/
https://ncbi.nlm.nih.gov/pubmed/29433126
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nature25478
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