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Mapping the Binding Trajectory of a Suicide Inhibitor in Human Indoleamine 2,3-Dioxygenase 1

Human indoleamine 2,3-dioxygenase 1 (hIDO1) is an important heme-containing enzyme that is a key drug target for cancer immunotherapy. Several hIDO1 inhibitors have entered clinical trials, among which BMS-986205 (BMS) stands out as the only suicide inhibitor. Despite its “best-in-class” activity, t...

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Podrobná bibliografie
Vydáno v:J Am Chem Soc
Hlavní autoři: Pham, Khoa N., Yeh, Syun-Ru
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6430111/
https://ncbi.nlm.nih.gov/pubmed/30347977
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.8b07994
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