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The mechanism of PI3Kα activation at the atomic level

PI3K lipid kinases phosphorylate PIP(2) to PIP(3) in the PI3K/Akt/mTOR pathway to regulate cellular processes. They are frequently mutated in cancer. Here we determine the PI3Kα activation mechanism at the atomic level. Unlike protein kinases where the substrate abuts the ATP, crystal structures ind...

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Bibliografiske detaljer
Udgivet i:Chem Sci
Main Authors: Zhang, Mingzhen, Jang, Hyunbum, Nussinov, Ruth
Format: Artigo
Sprog:Inglês
Udgivet: Royal Society of Chemistry 2019
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6430085/
https://ncbi.nlm.nih.gov/pubmed/30996962
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8sc04498h
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