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Discovery of New CDK8/CycC ligands with a Novel Virtual Screening Tool

Selective inhibition of Cyclin-dependent kinase 8 and cyclin C (CDK8/CycC) has been suggested as a promising strategy for reducing mitogenic signals in cancer cells with reduced toxic effects on normal cells. We developed a novel virtual screening protocol for drug development and applied it to disc...

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Dettagli Bibliografici
Pubblicato in:ChemMedChem
Autori principali: Chen, Wei, Ren, Xiaodong, Chang, Chia-en A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6428209/
https://ncbi.nlm.nih.gov/pubmed/30403831
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201800559
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