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Identification of Pyrazolo[1,5-a]pyridine-3-carboxamide Diaryl Derivatives as Drug Resistant Antituberculosis Agents

[Image: see text] A series of pyrazolo[1,5-a]pyridine-3-carboxamide (PPA) derivatives bearing diaryl side chain was designed and synthesized as new antituberculosis agents, aiming to improve the efficacy toward drug resistant Mycobacterium tuberculosis (Mtb) strains. Most of the substituted diphenyl...

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Detalhes bibliográficos
Publicado no:ACS Med Chem Lett
Main Authors: Hu, Xianglong, Wan, Baojie, Liu, Yang, Shen, Jiayi, Franzblau, Scott G., Zhang, Tianyu, Ding, Ke, Lu, Xiaoyun
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2019
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6421536/
https://ncbi.nlm.nih.gov/pubmed/30891129
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00410
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