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Identification of Pyrazolo[1,5-a]pyridine-3-carboxamide Diaryl Derivatives as Drug Resistant Antituberculosis Agents

[Image: see text] A series of pyrazolo[1,5-a]pyridine-3-carboxamide (PPA) derivatives bearing diaryl side chain was designed and synthesized as new antituberculosis agents, aiming to improve the efficacy toward drug resistant Mycobacterium tuberculosis (Mtb) strains. Most of the substituted diphenyl...

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Bibliografski detalji
Izdano u:ACS Med Chem Lett
Glavni autori: Hu, Xianglong, Wan, Baojie, Liu, Yang, Shen, Jiayi, Franzblau, Scott G., Zhang, Tianyu, Ding, Ke, Lu, Xiaoyun
Format: Artigo
Jezik:Inglês
Izdano: American Chemical Society 2019
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6421536/
https://ncbi.nlm.nih.gov/pubmed/30891129
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00410
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