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The atypical antipsychotic quetiapine induces hyperlipidemia by activating intestinal PXR signaling

Quetiapine, one of the most prescribed atypical antipsychotics, has been associated with hyperlipidemia and an increased risk for cardiovascular disease in patients, but the underlying mechanisms remain unknown. Here, we identified quetiapine as a potent and selective agonist for pregnane X receptor...

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Опубликовано в: :JCI Insight
Главные авторы: Meng, Zhaojie, Gwag, Taesik, Sui, Yipeng, Park, Se-Hyung, Zhou, Xiangping, Zhou, Changcheng
Формат: Artigo
Язык:Inglês
Опубликовано: American Society for Clinical Investigation 2019
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6413802/
https://ncbi.nlm.nih.gov/pubmed/30728326
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1172/jci.insight.125657
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