Wordt geladen...

Dithiocarbamate-inspired side chain stapling chemistry for peptide drug design

Two major pharmacological hurdles severely limit the widespread use of small peptides as therapeutics: poor proteolytic stability and membrane permeability. Importantly, low aqueous solubility also impedes the development of peptides for clinical use. Various elaborate side chain stapling chemistrie...

Volledige beschrijving

Bewaard in:
Bibliografische gegevens
Gepubliceerd in:Chem Sci
Hoofdauteurs: Li, Xiang, Tolbert, W. David, Hu, Hong-Gang, Gohain, Neelakshi, Zou, Yan, Niu, Fan, He, Wang-Xiao, Yuan, Weirong, Su, Jia-Can, Pazgier, Marzena, Lu, Wuyuan
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: Royal Society of Chemistry 2018
Onderwerpen:
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6357863/
https://ncbi.nlm.nih.gov/pubmed/30809370
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8sc03275k
Tags: Voeg label toe
Geen labels, Wees de eerste die dit record labelt!