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Efavirenz and Efavirenz-like Compounds Activate Human, Murine, and Macaque Hepatic IRE1α-XBP1

Efavirenz (EFV), a widely used antiretroviral drug, is associated with idiosyncratic hepatotoxicity and dyslipidemia. Here we demonstrate that EFV stimulates the activation in primary hepatocytes of key cell stress regulators: inositol-requiring 1α (IRE1α) and X-box binding protein 1 (XBP1). Followi...

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Publicat a:Mol Pharmacol
Autors principals: Heck, Carley J. S., Hamlin, Allyson N., Bumpus, Namandjé N.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2019
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6324649/
https://ncbi.nlm.nih.gov/pubmed/30442673
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.118.113647
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