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Spatial Distribution Profiles of Emtricitabine, Tenofovir, Efavirenz, and Rilpivirine in Murine Tissues Following In Vivo Dosing Correlate with Their Safety Profiles in Humans

[Image: see text] Emtricitabine (FTC), tenofovir (TFV), efavirenz (EFV), and rilpivirine (RPV) are currently used as components of HIV combination therapy. Although these drugs are widely used in antiretroviral therapy, several organ toxicities related to TFV and EFV have been observed clinically. T...

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Pubblicato in:ACS Pharmacol Transl Sci
Autori principali: Seneviratne, Herana Kamal, Hamlin, Allyson N., Heck, Carley J. S., Bumpus, Namandjé N.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2020
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7433710/
https://ncbi.nlm.nih.gov/pubmed/32832868
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsptsci.0c00015
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