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Discovery of 2-Piperidinyl Phenyl Benzamides and Trisubstituted Pyrimidines as Positive Allosteric Modulators of the Prostaglandin Receptor EP2

Prostaglandin E2 (PGE(2)) via its Gα(s)-coupled EP2 receptor protects cerebral cortical neurons from excitotoxic and anoxic injury, though EP2 receptor activation can also cause secondary neurotoxicity in chronic inflammation. We performed a high-throughput screen of a library of 292 000 small molec...

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Vydáno v:ACS Chem Neurosci
Hlavní autoři: Jiang, Jianxiong, Van, Tri Minh, Ganesh, Thota, Dingledine, Raymond
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6318807/
https://ncbi.nlm.nih.gov/pubmed/29292987
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.7b00486
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