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A conformationally-gated model of methadone and loperamide transport by P-glycoprotein

P-glycoprotein (Pgp) is a multidrug resistance transporter that limits the penetration of a wide range of neurotherapeutics into the brain including opioids. The diphenylpropylamine opioids methadone and loperamide are structurally similar, but loperamide has about a 4-fold higher Pgp-mediated trans...

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Vydáno v:J Pharm Sci
Hlavní autoři: Gibbs, Morgan E., Wilt, Laura A., Ledwitch, Kaitlyn V., Roberts, Arthur G.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6317893/
https://ncbi.nlm.nih.gov/pubmed/29499278
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.xphs.2018.02.019
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