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Celastrol induces ubiquitin-dependent degradation of mTOR in breast cancer cells

BACKGROUND: Celastrol is a major active component of the thunder god vine (Tripterygium wilfordii) used in traditional Chinese medicine to treat chronic inflammatory and autoimmune diseases. Celastrol inhibits PI3K–Akt–mTOR signaling, which is frequently dysregulated in tumors and critical for tumor...

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Dettagli Bibliografici
Pubblicato in:Onco Targets Ther
Autori principali: Li, Xiaoli, Zhu, Guangbei, Yao, Xintong, Wang, Ning, Hu, Ronghui, Kong, Qingxin, Zhou, Duanfang, Long, Liangyuan, Cai, Jiali, Zhou, Weiying
Natura: Artigo
Lingua:Inglês
Pubblicazione: Dove Medical Press 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6294079/
https://ncbi.nlm.nih.gov/pubmed/30588010
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/OTT.S187315
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