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Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms

The lack of efficacy of current antibacterials to treat multidrug resistant bacteria poses a life-threatening alarm. In order to develop enhancers of the antibacterial activity, we carried out a medicinal chemistry campaign aiming to develop inhibitors of enzymes that synthesise cysteine and belong...

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Detalhes bibliográficos
Publicado no:J Enzyme Inhib Med Chem
Main Authors: Magalhães, Joana, Franko, Nina, Annunziato, Giannamaria, Pieroni, Marco, Benoni, Roberto, Nikitjuka, Anna, Mozzarelli, Andrea, Bettati, Stefano, Karawajczyk, Anna, Jirgensons, Aigars, Campanini, Barbara, Costantino, Gabriele
Formato: Artigo
Idioma:Inglês
Publicado em: Taylor & Francis 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6217552/
https://ncbi.nlm.nih.gov/pubmed/30362368
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2018.1518959
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