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Histone Deacetylase 6-Selective Inhibitors and the Influence of Capping Groups on Hydroxamate-Zinc Denticity

Four crystal structures are presented of Histone Deacetylase 6 (HDAC6) complexes with para-substituted phenylhydroxamate inhibitors, including bulky peptoids. These structures provide insight regarding the design of capping groups that confer selectivity for binding to HDAC6, specifically with regar...

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Dades bibliogràfiques
Publicat a:J Med Chem
Autors principals: Porter, Nicholas J., Osko, Jeremy D., Diedrich, Daniela, Kurz, Thomas, Hooker, Jacob M., Hansen, Finn K., Christianson, David W.
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6136958/
https://ncbi.nlm.nih.gov/pubmed/30118224
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.8b01013
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