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Design, Synthesis and Biological Evaluation of 6,7-Disubstituted-4-phenoxyquinoline Derivatives Bearing Pyridazinone Moiety as c-Met Inhibitors

Deregulation of the receptor tyrosine kinase mesenchymal epithelial transition factor (MET) has been implicated in several human cancers and is an attractive target for small molecule drug discovery. Herein, a series of 6,7-disubstituted-4-phenoxyquinoline derivatives bearing pyridazinone derivative...

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Dades bibliogràfiques
Publicat a:Molecules
Autors principals: Liu, Xiaobo, Kou, Jianlan, Xiao, Zhen, Tian, Fajuan, Hu, Jiayi, Zheng, Pengwu, Zhu, Wufu
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6099740/
https://ncbi.nlm.nih.gov/pubmed/29949931
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules23071543
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