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Design, Synthesis and Biological Evaluation of 6,7-Disubstituted-4-phenoxyquinoline Derivatives Bearing Pyridazinone Moiety as c-Met Inhibitors

Deregulation of the receptor tyrosine kinase mesenchymal epithelial transition factor (MET) has been implicated in several human cancers and is an attractive target for small molecule drug discovery. Herein, a series of 6,7-disubstituted-4-phenoxyquinoline derivatives bearing pyridazinone derivative...

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Détails bibliographiques
Publié dans:Molecules
Auteurs principaux: Liu, Xiaobo, Kou, Jianlan, Xiao, Zhen, Tian, Fajuan, Hu, Jiayi, Zheng, Pengwu, Zhu, Wufu
Format: Artigo
Langue:Inglês
Publié: MDPI 2018
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6099740/
https://ncbi.nlm.nih.gov/pubmed/29949931
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules23071543
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