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Direct Imaging of Drug Distribution and Target Engagement of the PARP Inhibitor Rucaparib

Poly(ADP-ribose)polymerase (PARP) inhibitors have emerged as potent antitumor drugs. Here, we describe the intrinsic fluorescence properties of the clinically approved PARP inhibitor rucaparib and its potential to directly measure drug distribution and target engagement—a critical factor for underst...

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Dades bibliogràfiques
Publicat a:J Nucl Med
Autors principals: Kossatz, Susanne, Carney, Brandon, Farley, Christopher, Weber, Wolfgang A., Drain, Charles M., Reiner, Thomas
Format: Artigo
Idioma:Inglês
Publicat: Society of Nuclear Medicine 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6071506/
https://ncbi.nlm.nih.gov/pubmed/29572258
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2967/jnumed.117.205765
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