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Direct Imaging of Drug Distribution and Target Engagement of the PARP Inhibitor Rucaparib

Poly(ADP-ribose)polymerase (PARP) inhibitors have emerged as potent antitumor drugs. Here, we describe the intrinsic fluorescence properties of the clinically approved PARP inhibitor rucaparib and its potential to directly measure drug distribution and target engagement—a critical factor for underst...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:J Nucl Med
Egile Nagusiak: Kossatz, Susanne, Carney, Brandon, Farley, Christopher, Weber, Wolfgang A., Drain, Charles M., Reiner, Thomas
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Society of Nuclear Medicine 2018
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6071506/
https://ncbi.nlm.nih.gov/pubmed/29572258
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2967/jnumed.117.205765
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