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Direct Imaging of Drug Distribution and Target Engagement of the PARP Inhibitor Rucaparib

Poly(ADP-ribose)polymerase (PARP) inhibitors have emerged as potent antitumor drugs. Here, we describe the intrinsic fluorescence properties of the clinically approved PARP inhibitor rucaparib and its potential to directly measure drug distribution and target engagement—a critical factor for underst...

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Podrobná bibliografie
Vydáno v:J Nucl Med
Hlavní autoři: Kossatz, Susanne, Carney, Brandon, Farley, Christopher, Weber, Wolfgang A., Drain, Charles M., Reiner, Thomas
Médium: Artigo
Jazyk:Inglês
Vydáno: Society of Nuclear Medicine 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6071506/
https://ncbi.nlm.nih.gov/pubmed/29572258
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2967/jnumed.117.205765
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