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Deoxyschizandrin, a Naturally Occurring Lignan, Is a Specific Probe Substrate of Human Cytochrome P450 3A

To accurately predict the modifications done during metabolic processes by cytochrome P450 (P450) 3A enzyme, selecting substrates that best represent a broad range of substrate substitutions and that follow the Michaelis-Menten kinetic properties is highly necessary. In the present study, the oxidat...

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Publicat a:Drug Metab Dispos
Autors principals: Wu, Jingjing, Cao, Yunfeng, Zhang, Yanyan, Liu, Yong, Hong, James Y., Zhu, Liangliang, Ge, Guangbo, Yang, Ling
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6067378/
https://ncbi.nlm.nih.gov/pubmed/24131672
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.113.053884
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