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Novel VDR antagonists based on the GW0742 scaffold

The vitamin D receptor is a nuclear hormone receptor that regulates cell proliferation, cell differentiation and calcium homeostasis. The receptor is endogenously activated by 1,25-dihydroxyvitamin D(3), which induces transcription of VDR targets genes regulated by coactivator binding. VDR antagonis...

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Dades bibliogràfiques
Publicat a:Bioorg Med Chem Lett
Autors principals: Teske, Kelly A., Bogart, Jonathan W., Arnold, Leggy A.
Format: Artigo
Idioma:Inglês
Publicat: 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6008168/
https://ncbi.nlm.nih.gov/pubmed/29287957
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2017.12.041
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