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Beyond Competitive Inhibition: Regulation of ABC Transporters by Kinases and Protein-Protein Interactions as Potential Mechanisms of Drug-Drug Interactions

ATP-binding cassette (ABC) transporters are transmembrane efflux transporters mediating the extrusion of an array of substrates ranging from amino acids and lipids to xenobiotics, and many therapeutic compounds, including anticancer drugs. The ABC transporters are also recognized as important contri...

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Dettagli Bibliografici
Pubblicato in:Drug Metab Dispos
Autori principali: Crawford, Rebecca R., Potukuchi, Praveen K., Schuetz, Erin G., Schuetz, John D.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5896366/
https://ncbi.nlm.nih.gov/pubmed/29514827
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.118.080663
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