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Investigating the state dependence of drug binding in hERG channels using a trapped-open channel phenotype

The hERG channel is a key player in repolarization of the cardiac action potential. Pharmacological blockade of hERG channels depletes the cardiac repolarization reserve, increasing the risk of cardiac arrhythmias. The promiscuous nature of drug interactions with hERG presents a therapeutic challeng...

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Detalles Bibliográficos
Publicado en:Sci Rep
Main Authors: Thouta, Samrat, Lo, Garman, Grajauskas, Lukas, Claydon, Tom
Formato: Artigo
Idioma:Inglês
Publicado: Nature Publishing Group UK 2018
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5862968/
https://ncbi.nlm.nih.gov/pubmed/29563525
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-23346-x
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