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Structure-Based Design and Discovery of New M(2) Receptor Agonists

Muscarinic receptor agonists are characterized by apparently strict restraints on their tertiary or quaternary amine and their distance to an ester or related center. On the basis of the active state crystal structure of the muscarinic M(2) receptor in complex with iperoxo, we explored potential ago...

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Dettagli Bibliografici
Pubblicato in:J Med Chem
Autori principali: Fish, Inbar, Stößel, Anne, Eitel, Katrin, Valant, Celine, Albold, Sabine, Huebner, Harald, Möller, Dorothee, Clark, Mary J., Sunahara, Roger K., Christopoulos, Arthur, Shoichet, Brian K., Gmeiner, Peter
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5836741/
https://ncbi.nlm.nih.gov/pubmed/29094937
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.7b01113
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