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Design, semisynthesis and potent cytotoxic activity of novel 10-fluorocamptothecin derivatives

Fluorination is a well-known strategy for improving the bioavailability of bioactive molecules in the lead optimization phase of drug discovery projects. In an attempt to improve the antitumor activity of camptothecins (CPTs), novel 10-fluoro-CPT derivatives were designed, synthesized and evaluated...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Yang, Cheng-Jie, Song, Zi-Long, Goto, Masuo, Hsu, Pei-Ling, Zhang, Xiao-Shuai, Yang, Qian-Ru, Liu, Ying-Qian, Wang, Mei-Juan, Morris-Natschke, Susan L., Shang, Xiao-Fei, Lee, Kuo-Hsiung
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5831374/
https://ncbi.nlm.nih.gov/pubmed/28927790
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2017.09.012
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