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Oligo(lactic acid)(n)-paclitaxel prodrugs for poly(ethylene glycol)-block-poly(lactic acid) micelles: Loading, release and backbiting conversion for anticancer activity

Poly(ethylene glycol)-block-poly(D,L-lactic acid) (PEG-b-PLA) micelles are nanocarriers for poorly water-soluble anticancer agents and have advanced paclitaxel (PTX) into humans due to drug solubilization, biocompatibility and dose escalation. However, PEG-b-PLA micelles rapidly release PTX, resulti...

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Bibliografske podrobnosti
izdano v:J Am Chem Soc
Main Authors: Tam, Yu Tong, Gao, Jieming, Kwon, Glen S.
Format: Artigo
Jezik:Inglês
Izdano: 2016
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5576186/
https://ncbi.nlm.nih.gov/pubmed/27374999
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.6b03995
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