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Automated structure–activity relationship mining: connecting chemical structure to biological profiles

Understanding structure–activity relationships (SARs) of small molecules is important for developing probes and novel therapeutic agents in chemical biology and drug discovery. Increasingly multiplexed small-molecule profiling assays allow simultaneous measurement of many biological response paramet...

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Dettagli Bibliografici
Pubblicato in:J Biomol Screen
Autori principali: Wawer, Mathias J., Jaramillo, David E., Dancik, Vlado, Fass, Daniel M., Haggarty, Stephen J., Shamji, Alykhan F., Wagner, Bridget K., Schreiber, Stuart L., Clemons, Paul A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5554950/
https://ncbi.nlm.nih.gov/pubmed/24710340
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1177/1087057114530783
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