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A Single Amino Acid Residue at Transmembrane Domain 4 of the α Subunit Influences Carisoprodol Direct Gating Efficacy at GABA(A) Receptors

The muscle relaxant carisoprodol has recently been controlled at the federal level as a Schedule IV drug due to its high abuse potential and consequences of misuse, such as withdrawal syndrome, delusions, seizures, and even death. Recent work has shown that carisoprodol can directly gate and alloste...

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Détails bibliographiques
Publié dans:J Pharmacol Exp Ther
Auteurs principaux: Kumar, Manoj, Kumar, Manish, Freund, John M., Dillon, Glenn H.
Format: Artigo
Langue:Inglês
Publié: The American Society for Pharmacology and Experimental Therapeutics 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5539590/
https://ncbi.nlm.nih.gov/pubmed/28642232
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.117.242156
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