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Structure based discovery of new antagonist and biased agonist chemotypes for the Kappa Opioid Receptor

The ongoing epidemics of opioid overdose raises an urgent need for effective anti-addiction therapies and addiction-free painkillers. The κ–opioid receptor (KOR) has emerged as a promising target for both indications, raising demand for new chemotypes of KOR antagonists, as well as G-protein-biased...

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Bibliographische Detailangaben
Veröffentlicht in:J Med Chem
Hauptverfasser: Zheng, Zhong, Huang, Xi-Ping, Mangano, Thomas J., Zuo, Rodger, Chen, Xin, Zaidi, Saheem, Roth, Bryan L., Stevens, Raymond C., Katritch, Vsevolod
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2017
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5493393/
https://ncbi.nlm.nih.gov/pubmed/28339199
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.7b00109
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