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De Novo Modular Development of a Foldameric Protein–Protein Interaction Inhibitor for Separate Hot Spots: A Dynamic Covalent Assembly Approach

Protein–protein interactions stabilized by multiple separate hot spots are highly challenging targets for synthetic scaffolds. Surface‐mimetic foldamers bearing multiple recognition segments are promising candidate inhibitors. In this work, a modular bottom‐up approach is implemented by identifying...

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Pubblicato in:ChemistryOpen
Autori principali: Bartus, Éva, Hegedüs, Zsófia, Wéber, Edit, Csipak, Brigitta, Szakonyi, Gerda, Martinek, Tamás A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5390796/
https://ncbi.nlm.nih.gov/pubmed/28413758
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/open.201700012
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