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NMR-filtered virtual screening leads to non-metal chelating metallo-β-lactamase inhibitors

There are no clinically useful inhibitors of metallo-β-lactamases (MBLs), which are a growing problem because they hydrolyse almost all β-lactam antibacterials. Inhibition by most reported MBL inhibitors involves zinc ion chelation. A structure-based virtual screening approach combined with NMR filt...

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Bibliografski detalji
Izdano u:Chem Sci
Glavni autori: Li, Guo-Bo, Abboud, Martine I., Brem, Jürgen, Someya, Hidenori, Lohans, Christopher T., Yang, Sheng-Yong, Spencer, James, Wareham, David W., McDonough, Michael A., Schofield, Christopher J.
Format: Artigo
Jezik:Inglês
Izdano: Royal Society of Chemistry 2017
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5369532/
https://ncbi.nlm.nih.gov/pubmed/28451231
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6sc04524c
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