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Pharmacological targeting of BET proteins inhibits renal fibroblast activation and alleviates renal fibrosis

Bromodomain and extra-terminal (BET) protein inhibitors have been shown to effectively inhibit tumorgenesis and ameliorate pulmonary fibrosis by targeting bromodomain proteins that bind acetylated chromatin markers. However, their pharmacological effects in renal fibrosis remain unclear. In this stu...

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Dettagli Bibliografici
Pubblicato in:Oncotarget
Autori principali: Xiong, Chongxiang, Masucci, Monica V., Zhou, Xiaoxu, Liu, Na, Zang, Xiujuan, Tolbert, Evelyn, Zhao, Ting C., Zhuang, Shougang
Natura: Artigo
Lingua:Inglês
Pubblicazione: Impact Journals LLC 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5342478/
https://ncbi.nlm.nih.gov/pubmed/27732564
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.18632/oncotarget.12498
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