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Click chemistry reagent for identification of sites of covalent ligand incorporation in integral membrane proteins

Identifying sites of protein-ligand interaction is important for structure-based drug discovery and understanding protein structure-function relationships. Mass spectrometry (MS) has emerged as a useful tool for identifying residues covalently modified by ligands. Current methods use database search...

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Publicat a:Anal Chem
Autors principals: Budelier, Melissa M., Cheng, Wayland W. L., Bergdoll, Lucie, Chen, Zi-Wei, Abramson, Jeff, Krishnan, Kathiresan, Qian, Mingxing, Covey, Douglas F., Janetka, James W., Evers, Alex S.
Format: Artigo
Idioma:Inglês
Publicat: 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5328583/
https://ncbi.nlm.nih.gov/pubmed/28194953
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.analchem.6b05003
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