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Identification of allosteric binding sites for PI3Kα oncogenic mutant specific inhibitor design

PIK3CA , the gene that encodes the catalytic subunit of phosphatidylinositol 3-kinase α (PI3Kα), is frequently mutated in breast and other types of cancer. A specific inhibitor that targets the mutant forms of PI3Kα could maximize treatment efficiency while minimizing side-effects. Herein we describ...

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Bibliografische gegevens
Gepubliceerd in:Bioorg Med Chem
Hoofdauteurs: Miller, Michelle S., Maheshwari, Sweta, McRobb, Fiona M., Kinzler, Kenneth W., Amzel, L. Mario, Vogelstein, Bert, Gabelli, Sandra B.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2017
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5319926/
https://ncbi.nlm.nih.gov/pubmed/28129991
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2017.01.012
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