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Characterization of human cytochrome P450 mediated bioactivation of amodiaquine and its major metabolite N‐desethylamodiaquine

AIMS: Oxidative bioactivation of amodiaquine (AQ) by cytochrome P450s to a reactive quinoneimine is considered as an important mechanism underlying its idiosyncratic hepatotoxicity. However, because internal exposure to its major metabolite N‐desethylamodiaquine (DEAQ) is up to 240‐fold higher than...

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Detalhes bibliográficos
Publicado no:Br J Clin Pharmacol
Main Authors: Zhang, Yongjie, Vermeulen, Nico P. E., Commandeur, Jan N. M.
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5306493/
https://ncbi.nlm.nih.gov/pubmed/27718269
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcp.13148
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