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Charged propargyl-linked antifolates reveal mechanisms of antifolate resistance and inhibit trimethoprim-resistant MRSA strains possessing clinically relevant mutations

Drug-resistant enzymes must balance catalytic function with inhibitor destabilization to provide a fitness advantage. This sensitive balance, often involving very subtle structural changes, must be achieved through a selection process involving a minimal number of eligible point mutations. As part o...

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Bibliografische gegevens
Gepubliceerd in:J Med Chem
Hoofdauteurs: Reeve, Stephanie, Scocchera, Eric, Ferreira, Jacob, G-Dayanandan, Narendran, Keshipeddy, Santosh, Wright, Dennis L., Anderson, Amy C.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2016
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5257293/
https://ncbi.nlm.nih.gov/pubmed/27308944
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.6b00688
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