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Crystal structures of trimethoprim-resistant DfrA1 rationalize potent inhibition by propargyl-linked antifolates

Multidrug-resistant Enterobacteriaceae, notably Escherichia coli and Klebsiella pneumoniae, have become major health concerns worldwide. Resistance to effective therapeutics is often carried by class I and II integrons that can confer insensitivity to carbapenems, extended spectrum beta-lactamases,...

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Detalhes bibliográficos
Publicado no:ACS Infect Dis
Main Authors: Lombardo, Michael N., G-Dayanandan, Narendran, Wright, Dennis L., Anderson, Amy C.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5108240/
https://ncbi.nlm.nih.gov/pubmed/27624966
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.5b00129
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