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Inhibition of Antibiotic Efflux in Bacteria by the Novel Multidrug Resistance Inhibitors Biricodar (VX-710) and Timcodar (VX-853)

Inhibitors of mammalian multidrug efflux, such as the plant alkaloid reserpine, are also active in potentiating antibiotic activity by inhibiting bacterial efflux. Based on this precedent, two novel mammalian multiple drug resistance inhibitors, biricodar (VX-710) and timcodar (VX-853), were evaluat...

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Detalhes bibliográficos
Main Authors: Mullin, Steve, Mani, Nagraj, Grossman, Trudy H.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2004
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC525397/
https://ncbi.nlm.nih.gov/pubmed/15504837
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.48.11.4171-4176.2004
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