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Determination of the Kinetics and Thermodynamics of Ligand Binding to a Specific Inactive Conformation in Protein Kinases

Recent interest in inactive kinase conformations has generated the need to develop new biophysical tools to study them. Here, we describe the use of a fluorescent probe that selectively and potently binds to kinases in inactive, “DFG-out” conformations to obtain valuable thermodynamic and kinetic in...

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Pubblicato in:Methods Mol Biol
Autori principali: Hari, Sanjay B., Ranjitkar, Pratistha, Maly, Dustin J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5228460/
https://ncbi.nlm.nih.gov/pubmed/22956140
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/978-1-62703-008-3_12
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