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High-Affinity, Small-Molecule Peptidomimetic Inhibitors of MLL1/WDR5 Protein–Protein Interaction

Mixed lineage leukemia 1 (MLL1) is a histone H3 lysine 4 (H3K4) methyltransferase, and targeting the MLL1 enzymatic activity has been proposed as a novel therapeutic strategy for the treatment of acute leukemia harboring MLL1 fusion proteins. The MLL1/WDR5 protein–protein interaction is essential fo...

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Détails bibliographiques
Publié dans:J Am Chem Soc
Auteurs principaux: Karatas, Hacer, Townsend, Elizabeth C., Cao, Fang, Chen, Yong, Bernard, Denzil, Liu, Liu, Lei, Ming, Dou, Yali, Wang, Shaomeng
Format: Artigo
Langue:Inglês
Publié: 2012
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5180416/
https://ncbi.nlm.nih.gov/pubmed/23210835
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja306028q
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