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Identification of 1,2,3-triazole derivatives that protect pancreatic β cells against endoplasmmic reticulum stress-mediated dysfunction and death through the inhibition of C/EBP-homologous protein expression

The C/EBP-homologous protein (CHOP) acts as a mediator of endoplasmic reticulum (ER) stress-induced pancreatic insulin-producing β cell death, a key element in the pathogenesis of diabetes. Chemicals that inhibit the expression of CHOP might therefore protect β cells from ER stress-induced apoptosis...

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Dades bibliogràfiques
Publicat a:Bioorg Med Chem
Autors principals: Duan, Hongliang, Arora, Daleep, Li, Yu, Setiadi, Hendra, Xu, Depeng, Lim, Hui-Ying, Wang, Weidong
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5176337/
https://ncbi.nlm.nih.gov/pubmed/27157393
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2016.03.057
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